发明名称 NOVEL 3,4,4A,10B-TETRAHYDRO-1H-THIOPYRANO[4,3-C]ISOQUINOLINE COMPOUNDS
摘要 The compounds of formula (1) in which A, X, R1, R2, R3 and R7 have the meanings as given in the description, are novel effective inhibitors of type 4 and type 5 phosphodiesterase.
申请公布号 EP2721036(A1) 申请公布日期 2014.04.23
申请号 EP20120729458 申请日期 2012.06.12
申请人 TAKEDA GMBH 发明人 FLOCKERZI, DIETER;MANN, ALEXANDER;STENGEL, THOMAS;OHMER, HARALD;KAUTZ, ULRICH;WEINBRENNER, STEFFEN;FISCHER, STEFAN;TENOR, HERMANN;ZITT, CHRISTOF;HATZELMANN, ARMIN;DUNKERN, TORSTEN;HESSLINGER, CHRISTIAN;BRAUN, CLEMENS;BENEDIKTUS, EWALD;PAHL, ANDREAS;KÜLZER, RAIMUND;MARX, DEGENHARD
分类号 C07D495/04;A61K31/519;A61P11/00;C07D519/00 主分类号 C07D495/04
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