发明名称 |
Process for the preparation of aryl substituted olefinic amines |
摘要 |
An improved process for the preparation of aryl substituted olefinic amines such as (2S)-(4E)-N-methyl-5-[3-(5-isopropoxypyridin)yl]-4-penten-2-amine and (2S)-(4E)-N-methyl-5-[3-(5-methoxypyridin)yl]-4-penten-2-amine and new intermediates used in said process. |
申请公布号 |
US8703802(B2) |
申请公布日期 |
2014.04.22 |
申请号 |
US201113697807 |
申请日期 |
2011.05.19 |
申请人 |
DULL GARY MAURICE;GENUS JOHN;RATILAINEN TOMMI;RYBERG PER OLOF;HELLSTRÖM JANNA;WAHLSTRÖM NIKLAS;WÄNNMAN THOMAS;TARGACEPT, INC. |
发明人 |
DULL GARY MAURICE;GENUS JOHN;RATILAINEN TOMMI;RYBERG PER OLOF;HELLSTRÖM JANNA;WAHLSTRÖM NIKLAS;WÄNNMAN THOMAS |
分类号 |
A01N43/40;A61K31/435;A61K31/44;C07D213/62;C07D213/78 |
主分类号 |
A01N43/40 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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