发明名称 KINASE INHIBITORS AND METHODS OF USE THEREOF
摘要 The present invention provides compounds of formula I, pharmaceutically acceptable salts thereof, and pharmaceutical compositions thereof. Compounds of the present invention are useful for inhibiting kinase (e.g., GSK3 (e.g., GSK3αor GSK3β) or CK1) activity. The present invention further provides methods of using the compounds described herein for treating kinase-mediated disorders, such as neurological diseases, psychriatic disorders, metabolic disorders, and cancer.
申请公布号 US2014107141(A1) 申请公布日期 2014.04.17
申请号 US201314052661 申请日期 2013.10.11
申请人 WAGNER FLORENCE FEVRIER;PAN JENNIFER Q.;DANDAPANI SIVARAMAN;GERMAIN ANDREW;HOLSON EDWARD;MUNOZ BENITO;NAG PARTHA P.;WEIWER MICHEL;LEWIS MICHAEL C.;HAGGARTY STEPHEN J.;BISHOP JOSHUA A.;THE GENERAL HOSPITAL CORPORATION D/B/A MASSACHUSETTS GENERAL HOSPITAL;THE BROAD INSTITUTE, INC. 发明人 WAGNER FLORENCE FEVRIER;PAN JENNIFER Q.;DANDAPANI SIVARAMAN;GERMAIN ANDREW;HOLSON EDWARD;MUNOZ BENITO;NAG PARTHA P.;WEIWER MICHEL;LEWIS MICHAEL C.;HAGGARTY STEPHEN J.;BISHOP JOSHUA A.
分类号 C07D471/04;C07D471/10 主分类号 C07D471/04
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