发明名称 SYNTHESIS OF CHIRALLY PURIFIED SUBSTITUTED BENZOTHIAZOLE DIAMINES
摘要 Methods for preparing chirally purified substituted 4,5,6,7-tetrahydro-benzothiazole diamines such as, for example, (6R)2-amino-4,5,6,7-tetrahydro-6-(propylamino)benzothiazole and purifying a dominant enantiomer of substituted 4,5,6,7-tetrahydro-benzothiazole diamines from entantiomerically enriched mixtures of substituted 4,5,6,7-tetrahydro-benzothiazole diamines are provided herein.
申请公布号 US2014100372(A1) 申请公布日期 2014.04.10
申请号 US201313973987 申请日期 2013.08.22
申请人 KNOPP NEUROSCIENCES, INC. 发明人 RAJE PRASAD;GADIKOTA RAJENDRAKUMAR REDDY;CHEN JIAN-XIE;LAPINA OLGA V.;MCCALL JOHN M.
分类号 C07D277/82 主分类号 C07D277/82
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