发明名称 PROCESS FOR PRODUCING OPTICALLY ACTIVE SUCCINIMIDE DERIVATIVES AND INTERMEDIATES THEREOF
摘要 A process for producing optically active succinimide derivatives as key intermediates of (3R)-2′-(4-bromo-2-fluorobenzyl)spiro{pyrrolidine-3,4′(1′H)-pyrrolo[1,2-a]pyrazine}-1′,2,3′,5(2′H)-tetraone, which comprises the following reaction steps.
申请公布号 US2014099681(A1) 申请公布日期 2014.04.10
申请号 US201314104597 申请日期 2013.12.12
申请人 KYOWA HAKKO BIO CO., LTD.;DAINIPPON SUMITOMO PHARMA CO., LTD. 发明人 KASAI MASAJI;KITA SHINJI;OGAWA TADASHI;TOKAI HIDEAKI
分类号 C07D487/20;C12P17/18 主分类号 C07D487/20
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