发明名称 CRYSTALLINE FORM OF A QUINOLONE-CARBOXAMIDE COMPOUND
摘要 THE INVENTION PROVIDES A CRYSTALLINE HYDROCHLORIDE SALT OF 1-ISOPROPYL-2-OXO- 1,2-DIHYDROQUINOLINE-3-CARBOXYLIC ACID {(1,S,3R,5R)-8-[(R)-2-HYDROXY-3-(METHANESULFONYL-METHYL-AMINO)PROPYL]-8-AZABICYCLO[3.2.1]OCT-3-YL} AMIDE OR A SOLVATE THEREOF. THE INVENTION ALSO PROVIDES PHARMACEUTICAL COMPOSITIONS COMPRISING SUCH CRYSTALLINE SALT FORMS, METHODS OF USING SUCH CRYSTALLINE SALT FORMS TO TREAT DISEASES ASSOCIATED WITH 5-HT4 RECEPTOR ACTIVITY, AND PROCESSES USEFUL FOR PREPARING SUCH CRYSTALLINE SALT FORMS.
申请公布号 MY151075(A) 申请公布日期 2014.03.31
申请号 MY2006PI01482 申请日期 2006.04.03
申请人 THERAVANCE BIOPHARMA R&D IP, LLC 发明人 FATHEREE, PAUL R.;TURNER, S. DEREK;GOLDBLUM, ADAM, A.;CHAO, ROBERT;GENOV, DANIEL
分类号 C07D451/04 主分类号 C07D451/04
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