发明名称 |
CRYSTALLINE FORM OF A QUINOLONE-CARBOXAMIDE COMPOUND |
摘要 |
THE INVENTION PROVIDES A CRYSTALLINE HYDROCHLORIDE SALT OF 1-ISOPROPYL-2-OXO- 1,2-DIHYDROQUINOLINE-3-CARBOXYLIC ACID {(1,S,3R,5R)-8-[(R)-2-HYDROXY-3-(METHANESULFONYL-METHYL-AMINO)PROPYL]-8-AZABICYCLO[3.2.1]OCT-3-YL} AMIDE OR A SOLVATE THEREOF. THE INVENTION ALSO PROVIDES PHARMACEUTICAL COMPOSITIONS COMPRISING SUCH CRYSTALLINE SALT FORMS, METHODS OF USING SUCH CRYSTALLINE SALT FORMS TO TREAT DISEASES ASSOCIATED WITH 5-HT4 RECEPTOR ACTIVITY, AND PROCESSES USEFUL FOR PREPARING SUCH CRYSTALLINE SALT FORMS. |
申请公布号 |
MY151075(A) |
申请公布日期 |
2014.03.31 |
申请号 |
MY2006PI01482 |
申请日期 |
2006.04.03 |
申请人 |
THERAVANCE BIOPHARMA R&D IP, LLC |
发明人 |
FATHEREE, PAUL R.;TURNER, S. DEREK;GOLDBLUM, ADAM, A.;CHAO, ROBERT;GENOV, DANIEL |
分类号 |
C07D451/04 |
主分类号 |
C07D451/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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