发明名称 |
AMINOHETEROARYL COMPOUNDS AS PROTEIN KINASE INHIBITORS |
摘要 |
Aminopyridine and aminopyrazine compounds of formula (1), compositions including these compounds, and methods of their use are provided. Preferred compounds of formula 1 have activity as protein kinase inhibitors, including as inhibitors of c-MET. |
申请公布号 |
PL216368(B1) |
申请公布日期 |
2014.03.31 |
申请号 |
PL20040378759 |
申请日期 |
2004.02.26 |
申请人 |
SUGEN, INC. |
发明人 |
CUI JINGJONG JEAN;BHUMRALKAR DILIP;BOTROUS IRINY;CHU JI YU;FUNK LEE A.;HANAU CATHLEEN ELIZABETH;HARRIS G. DAVIS JR.;JIA LEI;JOHNSON JOANNE;KOLODZIEJ STEPHEN A.;KUNG PEI-PEI;LI XIAOYUAN(SHARON);LIN JASON(QISHEN);MENG JERRY JIALUN;NAMBU MITCHELL DAVID;NELSON CHRISTOPHER G.;PAIRISH MASON ALAN;SHEN HONG;TRAN-DUBE MICHELLE;WALTER ALLISON;ZHANG FANG-JIE;ZHANG JENNIFER |
分类号 |
C07D401/00;A61K;A61K31/44;A61K31/496;A61K31/4965;A61K31/497;C07D;C07D211/72;C07D213/73;C07D401/12;C07D403/00;C07D405/00;C07D409/00;C07D411/00;C07D413/00;C07D413/12;C07D417/00;C07D419/00 |
主分类号 |
C07D401/00 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|