发明名称 Processes and intermediates for making a JAK inhibitor
摘要 This invention relates to processes and intermediates for making {1-{1-[3-fluoro-2-(trifluoromethyl)isonicotinoyl]piperidin-4-yl}-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]azetidin-3-yl}acetonitrile, useful in the treatment of diseases related to the activity of Janus kinases (JAK) including inflammatory disorders, autoimmune disorders, cancer, and other diseases.
申请公布号 AU2012304650(A1) 申请公布日期 2014.03.27
申请号 AU20120304650 申请日期 2012.09.06
申请人 INCYTE CORPORATION 发明人 ZHOU, JIACHENG;LIU, PINGLI;CAO, GANFENG;WU, YONGZHONG
分类号 C07D487/04;C07D491/10 主分类号 C07D487/04
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