发明名称 REDUCTIVE AMINATION OF 6-KETO MORPHINANS BY CATALYTIC HYDROGEN TRANSFER
摘要 <p>The present invention provides compositions of 6-amino morphinan compounds and process for their synthesis. In particular, the processes provide for the reductive amination of 6-keto morphinans by catalytic transfer hydrogenation, to produce 6-amino morphinan compounds, which are epimerically and/or diastereomerically enriched.</p>
申请公布号 KR20140036215(A) 申请公布日期 2014.03.25
申请号 KR20137032225 申请日期 2012.06.08
申请人 MALLINCKRODT LLC 发明人 GROTE CHRISTOPHER W.;MCCLURG JOSEPH P.;JOHNSON JR. JOHN E.;FARRIS SARAH M.
分类号 C07D489/04;A61K31/485;A61P25/04 主分类号 C07D489/04
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