发明名称 BIPYRIDYLAMINOPYRIDINES AS SYK INHIBITORS
摘要 The present invention provides novel pyrimidine amines of formula I which are potent inhibitors of spleen tyrosine kinase, or are prodrugs thereof, and are useful in the treatment and prevention of diseases mediated by said enzyme, such as asthma, COPD and rheumatoid arthritis and cancer.
申请公布号 EP2706852(A1) 申请公布日期 2014.03.19
申请号 EP20120782391 申请日期 2012.05.04
申请人 MERCK SHARP & DOHME CORP.;MERCK CANADA INC. 发明人 DESCHENES, DENIS;ALTMAN, MICHAEL D.;ELLIS, JOHN MICHAEL;FISCHER, CHRISTIAN;HAIDLE, ANDREW M.;KATTAR, SOLOMON D.;NORTHRUP, ALAN B.;SCHELL, ADAM J.;SMITH, GRAHAM F.;TAOKA, BRANDON M.;BIENSTOCK, COREY;DI FRANCESCO, MARIA EMILIA;DONOFRIO, ANTHONY;PETERSON, SCOTT;SPENCER, KERRIE B.;JEWELL, JAMES PATRICK;ALI, AMJAD;BENNETT, DAVID JONATHAN;DANG, QUN;WAL, JOHN
分类号 A01N43/40;A61K31/44;C07D213/04 主分类号 A01N43/40
代理机构 代理人
主权项
地址