发明名称 SUBSTITUTED 3-CYANOQUINOLINES AS PROTEIN TYROSINE KINASES INHIBITORS
摘要 This invention provides compounds of formula 1 wherein R 1 , G 1 , G 2 , R 4 , Z, X and n are defined herein, or a pharmaceutically acceptable salt thereof, which are useful as antineoplastic agents and in the treatment of polycystic kidney disease.
申请公布号 EP2253620(B1) 申请公布日期 2014.03.12
申请号 EP20100173332 申请日期 1999.09.22
申请人 WYETH HOLDINGS LLC 发明人 WISSNER, ALLAN;TSOU, HWEI-RU;BERGER, DAN MAARTEN;FLOYD, MIDDLETON BRAWNER JR.;HAMANN, PHILIP ROSS;ZHANG, NAN;FROST, PHILIP
分类号 C07D215/54;A61K31/47;A61K31/4709;A61K31/496;A61K31/5377;A61K31/541;A61K31/553;A61P13/12;A61P35/00;C07D211/00;C07D215/56;C07D317/00;C07D401/04;C07D401/12;C07D405/12;C07D409/04;C07D413/12;C07D417/12;C07D491/10;C07D491/113;C07D521/00 主分类号 C07D215/54
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