发明名称 |
SUBSTITUTED 3-CYANOQUINOLINES AS PROTEIN TYROSINE KINASES INHIBITORS |
摘要 |
This invention provides compounds of formula 1
wherein R 1 , G 1 , G 2 , R 4 , Z, X and n are defined herein, or a pharmaceutically acceptable salt thereof, which are useful as antineoplastic agents and in the treatment of polycystic kidney disease. |
申请公布号 |
EP2253620(B1) |
申请公布日期 |
2014.03.12 |
申请号 |
EP20100173332 |
申请日期 |
1999.09.22 |
申请人 |
WYETH HOLDINGS LLC |
发明人 |
WISSNER, ALLAN;TSOU, HWEI-RU;BERGER, DAN MAARTEN;FLOYD, MIDDLETON BRAWNER JR.;HAMANN, PHILIP ROSS;ZHANG, NAN;FROST, PHILIP |
分类号 |
C07D215/54;A61K31/47;A61K31/4709;A61K31/496;A61K31/5377;A61K31/541;A61K31/553;A61P13/12;A61P35/00;C07D211/00;C07D215/56;C07D317/00;C07D401/04;C07D401/12;C07D405/12;C07D409/04;C07D413/12;C07D417/12;C07D491/10;C07D491/113;C07D521/00 |
主分类号 |
C07D215/54 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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