发明名称 HISTAMINE 4 RECEPTOR PARTIAL AGONISTS, INVERSE AGONISTS OR ANTAGONISTS FOR USE|IN TREATING NON-AUTOIMMUNE UVEITIS
摘要 The invention provides a compound which is a histamine 4 receptor antagonist, partial agonist or inverse agonist, for use in the treatment of non-autoimmune uveitis. The compound preferably has a structural core comprising a substituted pyrimidine group, such as an aminopyrimidine, diaminopyrimidine or triaminopyrimidine group, a thienopyrimidine, a furopyrimidine, a benzimidazole, an aryl or heteroaryl-fused pyrimidine, an indole, a bicyclic heteroaryl-substituted imidazole or a quinazoline group.
申请公布号 WO2014033480(A1) 申请公布日期 2014.03.06
申请号 WO2013GB52300 申请日期 2013.09.02
申请人 UCL BUSINESS PLC 发明人 CHALKIADAKIS, SPYRIDON;CALDER, VIRGINIA
分类号 A61K31/00;A61K31/454;A61K31/496;A61K31/506;A61K31/517;A61P27/02;G01N33/566 主分类号 A61K31/00
代理机构 代理人
主权项
地址