发明名称 BENZOXAZEPIN PI3K INHIBITOR COMPOUNDS AND THEIR USE IN THE TREATMENT OF CANCER
摘要 The invention relates to benzoxazepin compounds of Formula I including stereoisomers, geometric isomers, tautomers, or pharmaceutically acceptable salts thereof, wherein: Z 1 is CR 1 or N; Z 2 is CR 2 or N; Z 3 is CR 3 or N; Z 4 is CR 4 or N; and B is a pyrazolyl, imidazolyl, or triazolyl ring which compounds have anti-cancer activity, and more specifically, inhibit PI3 kinase activity.
申请公布号 PT2483278(E) 申请公布日期 2014.03.05
申请号 PT20100757213T 申请日期 2010.09.27
申请人 F. HOFFMANN-LA ROCHE AG 发明人 STEPHEN PRICE;ROBERT HEALD;NICOLE BLAQUIERE;STEVEN DO;DANETTE DUDLEY;ADRIAN J. FOLKES;TIMOTHY HEFFRON;MARK JONES;ALEKSANDR KOLESNIKOV;CHUDI NDUBAKU;ALAN G. OLIVERO;STEVEN STABEN;LAN WANG
分类号 C07D498/04;A61K31/4162;A61K31/4188;A61K31/4196;A61P35/00;C07D498/14;C07D519/00 主分类号 C07D498/04
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