发明名称
摘要 Ring-constrained amino acid surrogates of formula I where R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3</SUP>, R<SUP>4</SUP>, R<SUP>5</SUP>, R<SUP>6a</SUP>, R<SUP>6b</SUP>, R<SUP>7</SUP>, and y are as defined in the specification, methods for synthesizing ring-constrained amino acid surrogates of formula I, methods of use of ring-constrained amino acid surrogates of formula I, including use in linear or cyclic compounds which include a plurality of amino acid residues and one or more ring-constrained amino acid surrogates of formula I and linear or cyclic compounds which include a plurality of amino acid residues and one or more ring-constrained amino acid surrogates of formula I.
申请公布号 JP5424867(B2) 申请公布日期 2014.02.26
申请号 JP20090503307 申请日期 2007.03.30
申请人 发明人
分类号 C07D241/08;A61K38/22;A61P7/12;A61P9/04;A61P9/12;A61P13/02;A61P13/12;C07D243/08;C07D403/06;C07K7/00 主分类号 C07D241/08
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