发明名称 Crystalline form of a quinolinone-carboxamide compound
摘要 The invention provides a crystalline hydrochloride salt of 1-isopropyl-2-oxo-1,2-dihydroquinoline-3-carboxylic acid {(1S,3R,5R)-8-[(R)-2-hydroxy-3-(methanesulfonyl-methyl-amino)propyl]-8-azabicyclo[3.2.1]oct-3-yl}amide or a solvate thereof. The invention also provides pharmaceutical compositions comprising such crystalline salt forms, methods of using such crystalline salt forms to treat diseases associated with 5-HT4 receptor activity, and processes useful for preparing such crystalline salt forms.
申请公布号 US8658671(B2) 申请公布日期 2014.02.25
申请号 US20100759080 申请日期 2010.04.13
申请人 FATHEREE PAUL R.;TURNER S. DEREK;GOLDBLUM ADAM A.;CHAO ROBERT S.;GENOV DANIEL;THERAVANCE, INC. 发明人 FATHEREE PAUL R.;TURNER S. DEREK;GOLDBLUM ADAM A.;CHAO ROBERT S.;GENOV DANIEL
分类号 A61K31/46;C07D451/02 主分类号 A61K31/46
代理机构 代理人
主权项
地址