发明名称 PRODRUG DERIVATIVES OF (E)-N-METHYL-N-((3-METHYLBENZOFURAN-2-YL)METHYL)-3-(7-OXO-5,6,7,8-TETRAHYDRO-1,8-NAPHTHYRIDIN-3-YL)ACRYLAMIDE
摘要 In part, the present disclosure is directed to prodrug derivatives of (E)-N-methyl-N-((3-methylbenzofuran-2-yl)methyl)-3-(7-oxo-5,6,7,8-tetrahydro-1, 8-naphthyridin-3-yl)acrylamide compounds with significant solubility and bioavailability profiles.
申请公布号 US2014051666(A1) 申请公布日期 2014.02.20
申请号 US201314010166 申请日期 2013.08.26
申请人 AFFINIUM PHARMACEUTICALS, INC. 发明人 PARTRIDGE JOHN J.;COLUCCI JOHN;GAREAU YVES;THERIEN MICHEL;ZAMBONI ROBERT;HAFKIN BARRY;MARFAT ANTHONY;ZAGHDANE HELMI
分类号 C07F9/58;A61K31/675;A61K45/06 主分类号 C07F9/58
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