发明名称 |
PRODRUG DERIVATIVES OF (E)-N-METHYL-N-((3-METHYLBENZOFURAN-2-YL)METHYL)-3-(7-OXO-5,6,7,8-TETRAHYDRO-1,8-NAPHTHYRIDIN-3-YL)ACRYLAMIDE |
摘要 |
In part, the present disclosure is directed to prodrug derivatives of (E)-N-methyl-N-((3-methylbenzofuran-2-yl)methyl)-3-(7-oxo-5,6,7,8-tetrahydro-1, 8-naphthyridin-3-yl)acrylamide compounds with significant solubility and bioavailability profiles. |
申请公布号 |
US2014051666(A1) |
申请公布日期 |
2014.02.20 |
申请号 |
US201314010166 |
申请日期 |
2013.08.26 |
申请人 |
AFFINIUM PHARMACEUTICALS, INC. |
发明人 |
PARTRIDGE JOHN J.;COLUCCI JOHN;GAREAU YVES;THERIEN MICHEL;ZAMBONI ROBERT;HAFKIN BARRY;MARFAT ANTHONY;ZAGHDANE HELMI |
分类号 |
C07F9/58;A61K31/675;A61K45/06 |
主分类号 |
C07F9/58 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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