PROCESSES FOR THE PREPARATION OF (S)-3-4-((4-(MORPHOLINOMETHYL) BENZYL)OXY)-1-OXOISOINDOLIN-2-YL) PIPERIDINE-2,6-DIONE AND PHARMACEUTICALLY ACCEPTABLE FORMS THEREOF
摘要
Provided are processes for the preparation of enantiomerically enriched or enantiomerically pure 3-(4-((4-(morpholinomethyl)benzyl)oxy)- 1 -oxoisoindolin-2-yl)piperidine- 2,6-dione, or a pharmaceutically acceptable form thereof.
申请公布号
WO2014025978(A1)
申请公布日期
2014.02.13
申请号
WO2013US54099
申请日期
2013.08.08
申请人
CELGENE CORPORATION
发明人
TRAVERSE, JOHN, F.;ZHANG, CHENGMIN;FEIGELSON, GREGG, B.;COHEN, BENJAMIN, M.;LEONG, WILLIAM, W.