| 发明名称 |
N-CYCLOPROPYL-N-PIPERIDINYL-AMIDES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND USES THEREOF |
| 摘要 |
The present invention relates to compounds of general formula I, wherein R1, LP, HetAr1, (Het)Ar2 and n are as defined in the application, which have valuable pharmacological properties, and in particular bind to the GPR119 receptor and modulate its activity. |
| 申请公布号 |
US2014045823(A1) |
申请公布日期 |
2014.02.13 |
| 申请号 |
US201313955170 |
申请日期 |
2013.07.31 |
| 申请人 |
NOSSE BERND;ECKHARDT MATTHIAS;HIMMELSBACH FRANK;LANGKOPF ELKE;ASHWEEK NEIL J.;HARRIOTT NICOLE;NEUROCRINE BIOSCIENCES, INC.;BOEHRINGER INGELHEIM INTERNATIONAL GMBH |
发明人 |
NOSSE BERND;ECKHARDT MATTHIAS;HIMMELSBACH FRANK;LANGKOPF ELKE;ASHWEEK NEIL J.;HARRIOTT NICOLE |
| 分类号 |
C07D401/12;A61K31/454;A61K31/4545;A61K31/497;A61K31/506;A61K31/553;A61K45/06;C07D401/14;C07D413/12;C07D413/14 |
主分类号 |
C07D401/12 |
| 代理机构 |
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