发明名称 PROCESS FOR THE PREPARATION OF ANHYDROUS ARIPIPRAZOLE CRYSTAL FORM II
摘要 <p>The present invention relates to a process for preparation of aripiprazole crystal form II by recrystallizing aripiprazole in a mixture of acetone and 1-methoxy-2-propanol or a single solvent of 1-methoxy-2-propanol. The simple process according to the present invention can produce aripiprazole crystal form II with high purity and high yield in a mass scale.</p>
申请公布号 EP2691387(A2) 申请公布日期 2014.02.05
申请号 EP20120763355 申请日期 2012.03.30
申请人 DAEWOONG PHARMACEUTICAL CO., LTD. 发明人 CHOI, SOO JIN;OH, SEONG SOO;JIN, YONG SUK;KIM, YONG TAE;LEE, SEUNG JAE;SON, JEONG HYUN
分类号 C07D401/12;A61K31/4709;A61K31/496;A61P25/00;C07D215/227 主分类号 C07D401/12
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