INTERMEDIÁRIOS E PROCESSO ÚTIL NA PREPARAÇÃO DE {2-[1-(3,5-BIS-TRIFLUOROMETIL-BENZIL)-5-PIRIDIN-4-IL-1H[1,2, 3]TRIAZOL-4-IL]-PIRIDIN-3-IL}-2-CLOROFENIL)-METANONA

摘要

The present invention relates to novel compounds, (2-chlorophenyl)-[2-(2-hydroxy-2-pyridin-4-yl-vinyl)pyridin-3-yl]methanone benzoate, and (2-chlorophenyl)-[2-(2-hydroxy-2-pyridin-4-yl-vinyl)pyridin-3-yl]methanone toluate, which are useful intermediates for the preparation of the compound of Formula I: (I) The present invention further relates to novel processes for preparing a crystalline compound, which is {2-[1-(3,5-bis-trifluoromethyl-benzyl)-5-pyridin-4-yl-1H-[1,2,3]triazol-4-yl]-pyridin-3-yl}-(2-chlorophenyl)-methanone, Form IV.