发明名称 |
Antiviral compounds |
摘要 |
596444 Disclosed herein are anti-viral compounds, compositions containing such compounds, and the use of said compounds and compositions in the treatment of hepatitis C or a hepatitis C associated disorder, as well as to processes and intermediates useful for preparing such compounds. A preferred embodiment of the compound is (1-{ 3-[6-(9,9-difluoro-7-{ 2-[5-(2-methoxycarbonylamino-3-methylbutyryl)-5-aza-spiro[2.4]hept-6-yl]-3H-imidazol-4-yl} -9H-fluoren-2-yl)-1H-benzoimidazol-2-yl]-2-aza-bicyclo[2.2.1]heptane-2-carbonyl} -2-methyl-propyl)-carbamic acid methyl ester. |
申请公布号 |
NZ596444(A) |
申请公布日期 |
2014.01.31 |
申请号 |
NZ20100596444 |
申请日期 |
2010.05.12 |
申请人 |
GILEAD SCIENCES INC. |
发明人 |
COTTELL JEROMY J.;JIN HAOLUN;YANG ZHENG-YU;LIU QI;HALCOMB RANDALL L.;CANALES EDA;CHO AESOP;KIM CHOUNG U.;XU LIANHONG;PARRISH JAY P.;MISH MICHAEL R.;METOBO SAMUEL E.;DESAI MANOJ C.;KRYGOWSKI EVAN S.;SCHROEDER SCOTT D.;SHENG XIAONING;LAZERWITH SCOTT E.;SAUGIER JOSEPH H.;TSE WINSTON C.;VIVIAN RANDALL W.;GUO HONGYAN;PYUN HYUNG-JUNG;LIU HONGTAO;PHILLIPS BARTON W.;TAYLOR JAMES;BACON ELIZABETH M.;KATO DARRYL;LINK JOHN O.;CHOU CHIEN-HUNG;MCFADDEN RYAN;KELLAR TERRY;CLARKE MICHAEL O&rsquo,NEIL HANRAHAN;WATKINS WILLIAM J.;KIRSCHBERG THORSTEN A.;TRENKLE JAMES D.;MITCHELL MICHAEL L.;GRAUPE MICHAEL;VENKATARAMANI CHANDRASEKAR;SQUIRES NEIL;SUN JIANYU;MACKMAN RICHARD |
分类号 |
C07D401/14;C07D235/04;C07D403/04;C07D403/14;C07D405/14;C07D409/14;C07D413/04;C07D417/04;C07D417/14;C07D495/04 |
主分类号 |
C07D401/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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