发明名称 NOVEL CRYSTAL FORM OF 17α-ACETOXY-21-METOXY-11&bgr;-[4-N,N-DIMETHYLAMINOPHENYL]-19-NORPREGNA-4,9-DIENE-3,20-DIONE AND PROCESS FOR THE PREPARATION THEREOF
摘要 The present invention relates to novel crystalline Form II of 17α-acetoxy-21-methoxy-11&bgr;-[4-N,N-dimethylaminophenyl]-19-norpregna-4,9-diene-3,20-dione, (also known as CDB-4124), processes for the preparation thereof and pharmaceutical composition comprising it. Form II can be crystallized from different medium such as esters of C-Calcohols and carboxylic acids, ketones, cyclohexane, acetonitrile, dimethylformamide, dimethyl sulfoxide, water and any mixture thereof.
申请公布号 EA019114(B1) 申请公布日期 2014.01.30
申请号 EA20120000241 申请日期 2010.08.05
申请人 RICHTER GEDEON NYRT. 发明人 BALAZS ATTILA;CSOERGEI JANOS;DEMETER ADAM;SANTA CSABA
分类号 C07J41/00;A61K31/573;A61P5/36 主分类号 C07J41/00
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