发明名称 AZABICYCLIC CARBOXAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF
摘要 <p>THE INVENTION RELATES TO THE COMPOUNDS OF GENERAL FORMULA (I) IN WHICH X?, X?, X? AND X? ARE, INDEPENDENTLY OF ONE ANOTHER, A NITROGEN ATOM OR A C-R? GROUP; Z?, Z?, Z? AND Z? ARE, INDEPENDENTLY OF ONE ANOTHER, A NITROGEN ATOM OR A C-R? GROUP; Ra AND Rb FORM, TOGETHER WITH THE CARBON ATOMS WHICH BEAR THEM, A FIVE-MEMBERED RING, THIS RING COMPRISING A NITROGEN ATOM AND CARBON ATOMS, THIS RING BEING PARTIALLY SATURATED OR UNSATURATED AND BEING OPTIONALLY SUBSTITUTED WITH ONE OR MORE SUBSTITUENTS R?; W IS AN OXYGEN OR SULPHUR ATOM; n IS EQUAL TO 0, 1, 2 OR 3; Y IS AN OPTIONALLY SUBSTITUTED ARYL OR HETEROARYL; IN THE FORM OF A BASE OR OF AN ADDITION SALT WITH AN ACID, AND ALSO IN THE FORM OF A HYDRATE OR OF A SOLVATE. PROCESS FOR THE PREPARATION THEREOF AND THERAPEUTIC USE.</p>
申请公布号 MY150576(A) 申请公布日期 2014.01.30
申请号 MY2010PI03439 申请日期 2009.01.20
申请人 SANOFI-AVENTIS 发明人 DUBOIS LAURENT;EVANNO, YANNICK;MACHNIK DAVID;MALANDA, ANDRÉ
分类号 A61K31/4353 主分类号 A61K31/4353
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