摘要 |
<p>THE INVENTION RELATES TO THE COMPOUNDS OF GENERAL FORMULA (I) IN WHICH X?, X?, X? AND X? ARE, INDEPENDENTLY OF ONE ANOTHER, A NITROGEN ATOM OR A C-R? GROUP; Z?, Z?, Z? AND Z? ARE, INDEPENDENTLY OF ONE ANOTHER, A NITROGEN ATOM OR A C-R? GROUP; Ra AND Rb FORM, TOGETHER WITH THE CARBON ATOMS WHICH BEAR THEM, A FIVE-MEMBERED RING, THIS RING COMPRISING A NITROGEN ATOM AND CARBON ATOMS, THIS RING BEING PARTIALLY SATURATED OR UNSATURATED AND BEING OPTIONALLY SUBSTITUTED WITH ONE OR MORE SUBSTITUENTS R?; W IS AN OXYGEN OR SULPHUR ATOM; n IS EQUAL TO 0, 1, 2 OR 3; Y IS AN OPTIONALLY SUBSTITUTED ARYL OR HETEROARYL; IN THE FORM OF A BASE OR OF AN ADDITION SALT WITH AN ACID, AND ALSO IN THE FORM OF A HYDRATE OR OF A SOLVATE. PROCESS FOR THE PREPARATION THEREOF AND THERAPEUTIC USE.</p> |