发明名称 PROCESS FOR PREPARING ACYCLIC HCV PROTEASE INHIBITORS
摘要 Disclosed are highly convergent processes for preparing compounds of formula (I), which compounds are potent active agents for the treatment of hepatitis C virus (HCV) infection. The disclosed processes use SNAr-type coupling reactions between peptidic compounds having a hydroxyproline moiety and halogenated or sulfonated bromoquinoline compounds.
申请公布号 CA2568008(C) 申请公布日期 2014.01.28
申请号 CA20052568008 申请日期 2005.05.23
申请人 BOEHRINGER INGELHEIM INTERNATIONAL GMBH 发明人 BUSACCA, CARL ALAN;FRUTOS, ROGELIO PEREZ;HADDAD, NIZAR;KAPADIA, SURESH R.;LORENZ, JON CHARLES;SAHA, ANJAN;SENANAYAKE, CHRIS HUGH;WEI, XUDONG
分类号 C07K5/08;A61K31/4709;C07C217/84;C07C225/22;C07D277/56;C07D417/04;C07D417/14;C07K5/083 主分类号 C07K5/08
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