发明名称 NOVEL POLYMORPHS OF AZILSARTAN
摘要 <p>The present invention provides a novel crystalline form of azilsartan acid, process for its preparation and pharmaceutical compositions comprising it. The present invention also provides a novel crystalline form of azilsartan medoxomil potassium, process for its preparation and pharmaceutical compositions comprising it. Azilsartan medoxomil is chemically (5-methyl-2-oxo-1,3-dioxol-4-yl) methyl-2-ethoxy-1-([2'-(5-oxo-4,5-dihydro-1,2,4-oxadiazol-3-yl)biphenyl-4-yl]methyl)-1 H-benzimidazole-7-carboxylate. Azilsartan is an angiotensin II receptor antagonist used in the treatment of hypertension.</p>
申请公布号 CA2884248(A1) 申请公布日期 2014.01.16
申请号 CA20132884248 申请日期 2013.07.08
申请人 HETERO RESEARCH FOUNDATION 发明人 PARTHASARADHI REDDY, BANDI;RATHNAKAR REDDY, KURA;MURALIDHARA REDDY, DASARI;RAMAKRISHNA REDDY, MATTA;VAMSI KRISHNA, BANDI
分类号 C07D413/14;A61K31/4245 主分类号 C07D413/14
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