发明名称 |
NOVEL POLYMORPHS OF AZILSARTAN |
摘要 |
<p>The present invention provides a novel crystalline form of azilsartan acid, process for its preparation and pharmaceutical compositions comprising it. The present invention also provides a novel crystalline form of azilsartan medoxomil potassium, process for its preparation and pharmaceutical compositions comprising it. Azilsartan medoxomil is chemically (5-methyl-2-oxo-1,3-dioxol-4-yl) methyl-2-ethoxy-1-([2'-(5-oxo-4,5-dihydro-1,2,4-oxadiazol-3-yl)biphenyl-4-yl]methyl)-1 H-benzimidazole-7-carboxylate. Azilsartan is an angiotensin II receptor antagonist used in the treatment of hypertension.</p> |
申请公布号 |
CA2884248(A1) |
申请公布日期 |
2014.01.16 |
申请号 |
CA20132884248 |
申请日期 |
2013.07.08 |
申请人 |
HETERO RESEARCH FOUNDATION |
发明人 |
PARTHASARADHI REDDY, BANDI;RATHNAKAR REDDY, KURA;MURALIDHARA REDDY, DASARI;RAMAKRISHNA REDDY, MATTA;VAMSI KRISHNA, BANDI |
分类号 |
C07D413/14;A61K31/4245 |
主分类号 |
C07D413/14 |
代理机构 |
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代理人 |
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主权项 |
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