发明名称 ARIPIPRAZOLE-ORGANIC ACID COCRYSTAL, PREPARATION OR COMPOSITION CONTAINING SAME, AND PREPARATION METHOD THEREFOR
摘要 <p>The present invention relates to an aripiprazole-organic acid cocrystal in which aripiprazole and an organic acid form a cocrystal, a preparation or a composition containing the same, and a preparation method therefor. According to the present invention, it is possible to secure: a hygroscopicity-removed novel cocrystal by adding an organic acid such as salicylic acid and the like to aripiprazole anhydrous crystals; a convenient cocrystal preparation and the safety of a worker by developing a grinding method effective for industrialization; and a method for preparing a cocrystal capable of proceeding without a special chemical apparatus.</p>
申请公布号 WO2014003400(A1) 申请公布日期 2014.01.03
申请号 WO2013KR05574 申请日期 2013.06.25
申请人 GCB CO., LTD 发明人 AHN, SHINBYOUNG
分类号 C07D401/12;A61K9/00;A61K31/496 主分类号 C07D401/12
代理机构 代理人
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