发明名称 HCV PRODRUG FORMULATION
摘要 The present invention relates to a pharmaceutical composition comprising a solid suspension prepared by hot melt extrusion of isobutyric acid (2R,3S,4R,5R)-5-(4-amino-2-oxo-2H-pyrimidin-1-yl)-2-azido-3,4-bis-iso-butyryloxy-tetrahydro-furan-2-ylmethyl ester; hydrochloride salt (I) and a polyethylene glycol (PEG)/polypropylene glycol (PPG) block copolymer.
申请公布号 KR20080089344(A) 申请公布日期 2008.10.06
申请号 KR20087014073 申请日期 2008.06.12
申请人 F. HOFFMANN-LA ROCHE AG 发明人 AHMED HASHIM A.;ALFREDSON THOMAS VERNON;BIRUDARAJ KONDAMRAJ;BRANDL MICHAEL THOMAS;PHUAPRADIT WANTANEE;SHAH NAVNIT HARGOVINDAS;STEFANIDIS DIMITRIOS
分类号 A61K31/522;A61K9/16;A61K9/50;A61K31/506 主分类号 A61K31/522
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