发明名称 DERIVATIVES OF INDOLE-2-CARBOXAMIDES AND OF AZAINDOLE-2-CARBOXAMIDES SUBSTITUTED WITH A SILANYL GROUP, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF
摘要 THE INVENTION RELATES TO COMPOUNDS OF THE GENERAL FORMULA (I) IN WHICH: G?, G?, G? ET G? ARE INDEPENDENT FROM ONE ANOTHER, A C-X GROUP OR A NITROGEN ATOM; ONE OF G?, G?, G? AND G? AND AT MOST ONE OF G?, G?, G? AND G?IS A C-X GROUP IN WHICH X IS A -Si(X?)(X?)(X?) GROUP; N IS 0, 1, 2 OR 3; Y IS AN OPTIONALLY SUBSTITUTED ARYL OR HETEROARYL; ZI, Z2, Z3, Z4 ARE INDEPENDENT FROM ONE ANOTHER, A NITROGEN ATOM OR A C(R?) GROUP, AT LEAST ONE BEING A NITROGEN ATOM AND AT LEAST ONE BEING A C(R?) GROUP; Z IS CYCLIC AMINO OR ACYCLIC AMINO; SAID COMPOUNDS CAN BE IN THE STATE OF A BASE OR AN ADDITION SALT TO AN ACID, AS WELL AS IN THE HYDRATE OR SOLVATE STATE. THE INVENTION ALSO RELATES TO A METHOD FOR PREPARING THE SAME AND TO THE THERAPEUTIC USE THEREOF.
申请公布号 MY150289(A) 申请公布日期 2013.12.31
申请号 MY2010PI03446 申请日期 2009.01.20
申请人 SANOFI-AVENTIS 发明人 LAURENT DUBOIS;YANNICK EVANNO;ANDRE MALANDA
分类号 C07D401/12 主分类号 C07D401/12
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