发明名称 |
3-PYRAZIN SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AS JANUS KINASE INHIBITORS FOR THE TREATMENT OF CANCER DISEASES |
摘要 |
The present invention relates to pyrazine substituted pyrrolopyridines having formula (I) useful as inhibitors of JAK kinases (JAK1, JAK2, JAK3 and/or TYK2) and/or PDK1 and for the treatment of myeloproliferative disorders or other cancers. |
申请公布号 |
EP2211620(B1) |
申请公布日期 |
2013.12.25 |
申请号 |
EP20080841687 |
申请日期 |
2008.10.21 |
申请人 |
MERCK SHARP & DOHME CORP. |
发明人 |
GUERIN, DAVID, J.;JUNG, JOON;STANTON, ELIZABETH |
分类号 |
A01N43/90;A61K31/519;A61K31/535;C07D471/04 |
主分类号 |
A01N43/90 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|