发明名称 BENZODIAZEPINE DERIVATIVE FOR THE TREATMENT OF HEMATOPOIETIC NEOPLASM AND LEUKEMIA
摘要 <p>A method and medicament for treating mixed lineage leukemia; translocated mixed lineage leukemia; translocated mixed lineage leukemia based acute myelogenous leukemia; translocated mixed lineage leukemia based acute lymphoid leukemia; a non-MLL based chronic myeloproliferative disorder, or non-MLL based acute lymphoid leukemia is provided, wherein the active agent used is the GSK-3 inhibitor 7-(2,5-dihydro-4-imidazo[ 1,2-a]pyridine-3-yl-2,5-dioxo-1H-pyrrol-3-yl)-9-fluoro-1,2,3,4-tetrahydro-2-(1-piperidinylcarbonyl)-pyrrolo[3,2,1 jk][1,4]benzodiazepine or a pharmaceutically acceptable salt or solvate thereof.</p>
申请公布号 CA2758473(C) 申请公布日期 2013.12.17
申请号 CA20102758473 申请日期 2010.04.08
申请人 ELI LILLY AND COMPANY 发明人 CHEDID, MARCIO
分类号 A61K31/5517;A61P35/02 主分类号 A61K31/5517
代理机构 代理人
主权项
地址