| 发明名称 |
SYNTHESIS OF A VIRAL PROTEASE INHIBITOR |
| 摘要 |
<p>Disclosed is a process for the preparation of telaprevir of formula (I) or a salt thereof, comprising the oxidation reaction of a compound of formula (II) or a salt thereof, (II) wherein said oxidation is conducted in a solvent in the presence of a supported oxidising agent.</p> |
| 申请公布号 |
WO2013182636(A1) |
申请公布日期 |
2013.12.12 |
| 申请号 |
WO2013EP61681 |
申请日期 |
2013.06.06 |
| 申请人 |
DIPHARMA FRANCIS S.R.L. |
发明人 |
ALLEGRINI, PIETRO;BRUNOLDI, ENRICO;ATTOLINO, EMANUELE |
| 分类号 |
C07D403/12 |
主分类号 |
C07D403/12 |
| 代理机构 |
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代理人 |
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| 主权项 |
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| 地址 |
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