2-(4-OXO-4H-QUINAZOLIN-3-YL) ACETAMIDES AND THEIR USE AS VASOPRESSIN V3 ANTAGONISTS
摘要
The present invention relates to 2-(4-oxo4H-quinazolin-3-yl)acetamicle derivatives of formula (I), and to their use as vasopressin V3 antagonists, particularly for the treatment of depression.
申请公布号
CA2599511(C)
申请公布日期
2013.12.10
申请号
CA20062599511
申请日期
2006.03.10
申请人
N.V. ORGANON;PHARMACOPEIA DRUG DISCOVERY, INC.
发明人
LETOURNEAU, JEFFREY;RIVIELLO, CHRISTOPHER;HO, KOC-KAN;CHAN, JUI-HSIANG;OHLMEYER, MICHAEL;JOKIEL, PATRICK;NEAGU, IRINA;MORPHY, JOHN RICHARD;NAPIER, SUSAN ELIZABETH