发明名称 |
Moenomycin analogs, methods of synthesis, and uses thereof |
摘要 |
The present invention provides novel moenomycin analogs as well as pharmaceutical compositions thereof, methods of synthesis, and methods of use in treating an infection by administering an inventive compound to a subject in need thereof. The moenomycin analogs may be prepared synthetically, biosynthetically, or semi-synthetically. The analogs are particularly useful in treating or preventing infections caused by Gram-positive organisms. Certain inventive compounds may have a broader spectrum of coverage, which includes Gram-negative organisms. |
申请公布号 |
US8604004(B2) |
申请公布日期 |
2013.12.10 |
申请号 |
US20080681052 |
申请日期 |
2008.10.03 |
申请人 |
KAHNE DANIEL;KAHNE SUZANNE WALKER;ADACHI MASAATSU;DOUD EMMA;FUSE SHINICHIRO;LIN XIAONAN;ZHANG YI;TSUKAMOTO HIROKAZU;OSTASH BOHDAN;PRESIDENT AND FELLOWS OF HARVARD COLLEGE |
发明人 |
KAHNE DANIEL;KAHNE SUZANNE WALKER;ADACHI MASAATSU;DOUD EMMA;FUSE SHINICHIRO;LIN XIAONAN;ZHANG YI;TSUKAMOTO HIROKAZU;OSTASH BOHDAN |
分类号 |
A61K31/702;A61K31/7016;A61K31/7028;A61K31/715;C07H5/04;C07H5/06 |
主分类号 |
A61K31/702 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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