发明名称 |
PYRROLO[2,1-F][1,2,4]TRIAZINE COMPOUND, AND PREPARATION METHOD AND APPLICATION THEREOF |
摘要 |
<p>The present invention relates to a pyrrolo[2,1-f][1,2,4]triazine compound, an isomer thereof or a pharmaceutically acceptable salt, ester or hydrate thereof, and a preparation method and application thereof. The pyrrolo[2,1-f][1,2,4]triazine compound has a structure expressed in general formula (I). The pyrrolo[2,1-f][1,2,4]triazine compound expressed in general formula (I) can inhibit a phosphatidylinositol-3 kinase (PI3K) signal pathway, thereby being used to prepare medicine for treating phosphatidylinositol-3 kinase related diseases such as cancer.</p> |
申请公布号 |
CA2874062(A1) |
申请公布日期 |
2013.12.05 |
申请号 |
CA20132874062 |
申请日期 |
2013.04.23 |
申请人 |
SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES;SHANGHAI HAIHE PHARMACEUTICAL CO., LTD. |
发明人 |
YANG, CHUNHAO;MENG, LINGHUA;CHEN, YANHONG;WANG, XIANG;TAN, CUN;LI, JIAPENG;DING, JIAN;CHEN, YI |
分类号 |
C07D487/04;A61K31/5377;A61K31/5386;A61P35/00;C07D519/00 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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