发明名称 |
Process for preparing a 2-alkynyl substituted 5-amino-pyrazolo-[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine |
摘要 |
A process for preparing 7-[2-[4-(6-fluoro-3-methyl-1,2-benzisoxazol-5-yl)-1-piperazinyl]ethyl]-2-(1-propynyl)-7H-pyrazolo-[4,3-e]-[1,2,4]-triazolo[1,5-c]pyrimidin-5-amine, intermediates useful in that process, and processes for preparing said intermediates are disclosed. |
申请公布号 |
US8598343(B2) |
申请公布日期 |
2013.12.03 |
申请号 |
US201013389029 |
申请日期 |
2010.08.03 |
申请人 |
KUO SHEN-CHUN;CHEN YONGGANG;ECKERT JEFFREY M.;LEONG WILLIAM W.;ZOU NANFEI;KUKLIS GABRIEL C.;MERCK SHARP & DOHME CORP. |
发明人 |
KUO SHEN-CHUN;CHEN YONGGANG;ECKERT JEFFREY M.;LEONG WILLIAM W.;ZOU NANFEI;KUKLIS GABRIEL C. |
分类号 |
C07D491/00 |
主分类号 |
C07D491/00 |
代理机构 |
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