发明名称 HIGH DRUG LOAD TABLET FORMULATION OF BRIVANIB ALANINATE
摘要 The present invention is directed to a high drug load tablet formulation of [(1R), 2S]-2-aminopropionic acid 2-[4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy]-1-methylethyl ester, and to methods of using the formulation in the treatment of cancer.
申请公布号 EP2663283(A1) 申请公布日期 2013.11.20
申请号 EP20120702349 申请日期 2012.01.13
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 NARANG, AJIT S.;BADAWY, SHERIF IBRAHIM FARAG;SUBRAMANIAN, GANESHKUMAR A.;LAMARCHE, KEIRNAN RYAN;BINDRA, DILBIR S.;RAO, VENKATRAMANA M.
分类号 A61K9/00;A61K9/20;A61K9/28;A61K31/53;A61K47/02;A61K47/12;A61K47/26;A61K47/32;A61K47/36;A61K47/38;A61P35/00 主分类号 A61K9/00
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