发明名称 |
HIGH DRUG LOAD TABLET FORMULATION OF BRIVANIB ALANINATE |
摘要 |
The present invention is directed to a high drug load tablet formulation of [(1R), 2S]-2-aminopropionic acid 2-[4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy]-1-methylethyl ester, and to methods of using the formulation in the treatment of cancer. |
申请公布号 |
EP2663283(A1) |
申请公布日期 |
2013.11.20 |
申请号 |
EP20120702349 |
申请日期 |
2012.01.13 |
申请人 |
BRISTOL-MYERS SQUIBB COMPANY |
发明人 |
NARANG, AJIT S.;BADAWY, SHERIF IBRAHIM FARAG;SUBRAMANIAN, GANESHKUMAR A.;LAMARCHE, KEIRNAN RYAN;BINDRA, DILBIR S.;RAO, VENKATRAMANA M. |
分类号 |
A61K9/00;A61K9/20;A61K9/28;A61K31/53;A61K47/02;A61K47/12;A61K47/26;A61K47/32;A61K47/36;A61K47/38;A61P35/00 |
主分类号 |
A61K9/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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