发明名称 GPBP inhibition using Q2 peptidomimetics
摘要 Disclosed are compounds of formula: that inhibiting GPBP activity, making them useful as therapeutics in antibody-mediated disorders, drug-resistant cancer, inflammation, protein misfolding and ER stress-mediated disorders, and aberrant apoptosis.
申请公布号 US8586776(B2) 申请公布日期 2013.11.19
申请号 US20100940598 申请日期 2010.11.05
申请人 SAUS JUAN;FUSTERO SANTOS;SANZ-CERVERA JUAN F.;PEREZ-PAYA ENRIQUE;BLASCO RAUL;REVERT-ROS FRANCISCO;REVERT FERNANDO;FIBROSTATIN, S.L. 发明人 SAUS JUAN;FUSTERO SANTOS;SANZ-CERVERA JUAN F.;PEREZ-PAYA ENRIQUE;BLASCO RAUL;REVERT-ROS FRANCISCO;REVERT FERNANDO
分类号 C07C69/95 主分类号 C07C69/95
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