发明名称 |
GPBP inhibition using Q2 peptidomimetics |
摘要 |
Disclosed are compounds of formula: that inhibiting GPBP activity, making them useful as therapeutics in antibody-mediated disorders, drug-resistant cancer, inflammation, protein misfolding and ER stress-mediated disorders, and aberrant apoptosis.
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申请公布号 |
US8586776(B2) |
申请公布日期 |
2013.11.19 |
申请号 |
US20100940598 |
申请日期 |
2010.11.05 |
申请人 |
SAUS JUAN;FUSTERO SANTOS;SANZ-CERVERA JUAN F.;PEREZ-PAYA ENRIQUE;BLASCO RAUL;REVERT-ROS FRANCISCO;REVERT FERNANDO;FIBROSTATIN, S.L. |
发明人 |
SAUS JUAN;FUSTERO SANTOS;SANZ-CERVERA JUAN F.;PEREZ-PAYA ENRIQUE;BLASCO RAUL;REVERT-ROS FRANCISCO;REVERT FERNANDO |
分类号 |
C07C69/95 |
主分类号 |
C07C69/95 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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