发明名称 1,2,3,4-TETRAHYDROQUINOXALINE COMPOUNDS HAVING GLUCOCORTICOID RECEPTOR BINDING ACTIVITY
摘要 A 1,2,3,4-tetrahydroquinoxaline compound represented by the following formula: In the formula (1), R1 represents substituents such as a halogen, an alkyl, a cycloalkyl, an aryl or a heterocyclic group; p represents 0 to 5; R2 represents substituents such as a halogen, an alkyl, a hydroxyl or an alkoxy group; q represents 0 to 2; R3 represents substituents such as hydrogen, an alkyl, an alkenyl, an alkylcarbonyl or an arylcarbonyl group; R4 and R5 independently represent substituents such as hydrogen, a halogen, an alkyl, an alkenyl, an alkynyl, a cycloalkyl, an aryl or a heterocyclic group; R6 represents substituents such as hydrogen, an alkyl, an alkenyl, an alkynyl, a cycloalkyl, an aryl or a heterocyclic group; A represents an alkylene; R7 represents OR8, NR8R9, SR8, S(O)R8, S(O)2R8; R8 and R9 independently represent substituents such as hydrogen, an alkyl or an alkenyl; and X represents O or S.
申请公布号 US2013303537(A1) 申请公布日期 2013.11.14
申请号 US201313937447 申请日期 2013.07.09
申请人 SANTEN PHARMACEUTICAL CO., LTD. 发明人 MATSUDA MAMORU;MORI TOSHIYUKI;KAWASHIMA KENJI;YAMAMOTO MINORU;KATO MASATOMO;TAKAI MIWA;NAGATSUKA MASATO;KOBAYASHI SACHIKO
分类号 C07D241/46;C07D401/12;C07D405/12;C07D409/12;C07D409/14 主分类号 C07D241/46
代理机构 代理人
主权项
地址