发明名称 2-(6-HYDROXYMETHYL-9-METHYL-2-(2'-METHOXYPHENYL)-5H-PYRIDO[4',3':5,6]PYRANO[2,3-d]PYRIMIDINE-4-YLSULFANYL)ACETAMIDE WITH ANTIFUNGAL ACTIVITY
摘要 The invention relates to pyrido[4',3':5,6]pyrano[2,3-d] pyrimidine derivatives exhibiting antifungal activity against wide variety of Candida spp. cultures, including clinical isolates resistant to fluconazole such as C. albicans, C. famata, C. kefyr, C. pseudotropicalis, C. Rugosa, as well as aspergillosis and dermathophyte agents.
申请公布号 UA103638(C2) 申请公布日期 2013.11.11
申请号 UA20110007115 申请日期 2011.06.06
申请人 “MECHNYKOV INSTITUTE FOR MICROBIOLOGY AND IMMUNOLOGY OF AMS OF UKRAINE” STATE INSTITUTION 发明人 SCHERBAK OLHA MYKOLAIVNA;KUCHMA IRYNA YURIIVNA;KAZMIRCHYK VIKTOR VOLODYMYROVYCH;RUSAK PETRO STEPANOVYCH;ZHURAVEL` IRYNA OLEKSANDRIVNA;KRESTETSKA SVITLANA LEONIDIVNA;ANDREEVA IRYNA DMYTRIVNA;MYRONENKO LIUDMYLA HRYHORIVNA;VOLKOV TARAS OLEKSANDROVYCH;LAKHMAN SERHII MYKHAILOVYCH;CHERNYSHENKO DMYTRO MYKOLAIOVYCH;SHULHA NATALIA MYKOLAIVNA;PICHEVSKA NATALIA IVANIVNA;HOLUBKA OLHA VADYMIVNA;MAKARENKO VALENTYNA DMYTRIVNA
分类号 C07D491/147;A61K31/33 主分类号 C07D491/147
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