发明名称 |
PYRROLIDINONES AS METAP-2 INHIBITORS |
摘要 |
Compounds of the formula I in which R1, R2, R3 and R4 have the meanings indicated in Claim 1, are inhibitors of methionine aminopeptidase and can be employed for the treatment of tumours.
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申请公布号 |
US2013296274(A1) |
申请公布日期 |
2013.11.07 |
申请号 |
US201113878574 |
申请日期 |
2011.09.14 |
申请人 |
HEINRICH TIMO;ZENKE FRANK;CALDERINI MICHEL;MUSIL DJORDJE;MERCK PATENT GMBH |
发明人 |
HEINRICH TIMO;ZENKE FRANK;CALDERINI MICHEL;MUSIL DJORDJE |
分类号 |
C07D401/14;A61K31/4025;A61K31/422;A61K31/4245;A61K31/433;A61K31/4439;A61K31/4709;A61K31/5377;A61K31/69;A61K45/06;C07D401/10;C07D409/12;C07D413/12;C07F5/02 |
主分类号 |
C07D401/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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