发明名称 Pyridine-3-carboxyamide derivative
摘要 To provide a novel JAK3 inhibitor that is useful as a preventive and/or therapeutic agent for rejection and graft versus host disease (GvHD) in organ transplantation, rheumatoid arthritis, multiple sclerosis, systemic lupus erythematosus, Sjögren syndrome, Behcet's disease, type I diabetes mellitus, autoimmune thyroiditis, idiopathic thrombocytopenic purpura, ulcerative colitis, Crohn's disease, asthma, allergic rhinitis, atopic dermatitis, contact dermatitis, urticaria, eczema, psoriasis, allergic conjunctivitis, uveitis, cancer, leukemia and the like. The pyridine-3-carboxyamide derivative represented by the general formula (1): or its salt or a solvate thereof.
申请公布号 US8575153(B2) 申请公布日期 2013.11.05
申请号 US200913131561 申请日期 2009.11.27
申请人 KITAMURA TAKAHIRO;YAMADA HAJIME;TAKEMURA SHUNJI;ASHIKAWA MASANORI;ISHIKAWA TETSUYA;MIYAKE YOSHIHARU;KOUKETSU AKIYASU;SATO SEIICHI;ISHIWATA HIROYUKI;TABUNOKI YUICHIRO;SHIBASAKI MANABU;OZAWA TAKATOSHI;SHIGEMI RYOTA;DOI TAKESHI;TAMURA MASAHIRO;KOWA COMPANY, LTD. 发明人 KITAMURA TAKAHIRO;YAMADA HAJIME;TAKEMURA SHUNJI;ASHIKAWA MASANORI;ISHIKAWA TETSUYA;MIYAKE YOSHIHARU;KOUKETSU AKIYASU;SATO SEIICHI;ISHIWATA HIROYUKI;TABUNOKI YUICHIRO;SHIBASAKI MANABU;OZAWA TAKATOSHI;SHIGEMI RYOTA;DOI TAKESHI;TAMURA MASAHIRO
分类号 A61K31/506;C07D239/48 主分类号 A61K31/506
代理机构 代理人
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