发明名称 |
ACID ADDITION SALTS OF THE 2-[2-[[(4-METHOXY-2,6-DIMETHYLPHENYL)SULFONYL]-(METHYL)AMINO]ETHOXY]-N-METHYL-N-[3-(4-METHYLPIPERAZIN-1-YL)CYCLOHEXYL] ACETAMIDE AND THE USE THEREOF AS BRADYKININ B1 RECEPTORANTAGONISTS |
摘要 |
The present invention relates to the new acid addition salts AB of the following free base of formula A or the enantiomer thereof with a physiologically acceptable acid B which is selected from among hydrochloric acid, fumaric acid and tartaric acid, as well as the polymorphs, hydrates and solvates thereof.
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申请公布号 |
US2013289049(A1) |
申请公布日期 |
2013.10.31 |
申请号 |
US201113814006 |
申请日期 |
2011.08.04 |
申请人 |
PACHUR THORSTEN;PFRENGLE WALDEMAR;BIRK MANFRED;SCHNAUBELT JUERGEN;WERTHMANN ULRIKE;BOEHRINGER INGELHEIM INTERNATIONAL GMBH |
发明人 |
PACHUR THORSTEN;PFRENGLE WALDEMAR;BIRK MANFRED;SCHNAUBELT JUERGEN;WERTHMANN ULRIKE |
分类号 |
C07D295/155 |
主分类号 |
C07D295/155 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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