发明名称 |
PROCESS FOR PREPARING AMINO CROTONYL COMPOUNDS |
摘要 |
THE INVENTION RELATES TO AN IMPROVED PROCESS FOR PREPARING 4-[(3-CHLORO-4-FLUOROPHENYL)AMINO]-6-{[4-(N,N-DIMETHYLAMINO)-1-OXO-2-BUTEN-1-YL]AMINO}-7-((S)-TETRAHYDROFURAN-3-YLOXY)-QUINAZOLINE AND RELATED AMINOCROTONYL COMPOUNDS AND THE PREPARATION OF A SUITABLE SALT OF 4-[(3-CHLORO-4-FLUOROPHENYL)AMINO]-6-{[4-(N,N-DIMETHYLAMINO)-1-OXO-2-BUTEN-1-YL]AMINO}-7-((S)-TETRAHYDROFURAN-3-YLOXY)-QUINAZOLINE FOR USE AS A PHARMACEUTICALLY ACTIVE SUBSTANCE. |
申请公布号 |
MY149921(A) |
申请公布日期 |
2013.10.31 |
申请号 |
MY2004PI04237 |
申请日期 |
2004.10.14 |
申请人 |
BOEHRINGER INGELHEIM INTERNATIONAL GMBH |
发明人 |
RAINER SOYKA;WERNER RALL;JUERGEN SCHNAUBELT;PETER SIEGER;CHRISTIAN KULINNA |
分类号 |
C07D405/12;A61K31/505;A61K31/517 |
主分类号 |
C07D405/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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