发明名称 PROCESS FOR THE PREPARATION OF 2-(TRIAZINYLCARBONYL)SULFONANILIDES
摘要 The invention relates to a method, which is based on the oxidative ring opening of a compound with an oxindole structure, for producing substituted 2-(triazinylcarbonyl) sulfonanilides of formula (1-1) proceeding from an N-sulfonyl-substituted 3-triazinyl oxindole of formula (2-1), to the thus produced 2-(triazinylcarbonyl) sulfonanilides of formula (1-1), and to the use thereof as intermediate products for the synthesis of fine chemicals and active substances in the agricultural field. Furthermore, the invention relates to a multistage method for producing N-alkyl-N-[2-(1,3,5-triazin-2-ylcarbonyl)phenyl]alkansulfonamides of formula (4-1) proceeding from a 3-(alkylsulfanyl)-1,3-dihydro-2H-indol-2-on of formula (7-1), wherein the multistage method also has said oxidative opening as a sub-step, and to the 2-(triazinylcarbonyl) sulfonanilides of formula (1-1), said sulfonanilides being obtained by means of the oxidative ring opening and used as intermediates in the multistage method.
申请公布号 EP2655346(A2) 申请公布日期 2013.10.30
申请号 EP20110807678 申请日期 2011.12.19
申请人 BAYER INTELLECTUAL PROPERTY GMBH 发明人 KARIG, GUNTER;FORD, MARK, JAMES;SIEGEL, KONRAD
分类号 C07D251/20;A01N43/66;C07D403/04 主分类号 C07D251/20
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