BOMBESIN ANALOG PEPTIDE ANTAGONIST CONJUGATES

摘要

To provide a diagnostic and therapeutic medicament, a bombesin analog peptide antagonist conjugate is provided which has general Formula (I): [A-(B)]-C, wherein A is a metal chelator comprising at least one radionuclidc metal, B is a spacer linked to N-terminal of C or a covalent bond and C is a bombesin analog peptide antagonist having a sequence as claimed, where further x is an integer from 1 to 3 and n is an integer from 1 to 6.