发明名称 |
ISOTHIAZOLE-PYRIDINE DERIVATIVES AS MODULATORS OF HIF (HYPOXIA INDUCIBLE FACTOR) ACTIVITY |
摘要 |
<p>The present invention relates to novel compounds according to Formula I or II, methods, and compositions capable of decreasing HIF hydroxylase enzyme activity, thereby increasing the stability and/or activity of hypoxia inducible factor (HIF). Formula (I) or (II).</p> |
申请公布号 |
EP2252619(B1) |
申请公布日期 |
2013.10.09 |
申请号 |
EP20090700287 |
申请日期 |
2009.01.12 |
申请人 |
FIBROGEN, INC. |
发明人 |
ZHOU, XIAOTI;AREND, MICHAEL, P.;WU, MIN;FLIPPIN, LEE, A. |
分类号 |
C07D513/04;A61K31/4353;A61P9/00 |
主分类号 |
C07D513/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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