发明名称 METHOD FOR THE PREPARATION OF HIGH-PURITY PHARMACEUTICAL INTERMEDIATES
摘要 The present invention is related to intermediates useful in the preparation of pharmaceutically acceptable salts of (+)-7-[4-(4-fluorophenyl)-6-isopropyl-2-(methanesulfonyl-methyl-amino)-pyrimidin-5-yl]-(3R,5S)-dihydroxy-hept-6-enoic acid and polymorphs of said intermediates, methods for preparation thereof and use thereof.
申请公布号 EP2646420(A1) 申请公布日期 2013.10.09
申请号 EP20110819001 申请日期 2011.11.29
申请人 EGIS GYOGYSZERGYAR NYILVANOSAN MUEKOEDOE RESZVENYTARSASAG 发明人 KOVANYINE LAX, GYOERGYI;SIMIG, GYULA;VOLK, BALAZS;BARTHA, FERENC LORANT;KRASZNAI, GYOERGY;RUZSICS, GYOERGY;SIPOS, EVA;NAGY, KALMAN;MOROVJAN, GYOERGY;BARKOCZY, JOZSEF;KESZTHELYI, ADRIENN;IMRE, JANOS;BAGYINSZKI, GABOR
分类号 C07D239/42;A61K31/505 主分类号 C07D239/42
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