发明名称 |
PREPARATION OF NUCLEOSIDES RIBOFURANOSYL PYRIMIDINES |
摘要 |
The present process provides an improved method for the preparation of 4-amino-1-((2R,3R,4R,5R)-3-fluoro-4-hydroxy-5-hydrox-ymethyl-3-methyl-tetrahydro-furan-2-yl)-1H-pyrimidin-2-one of the formula (IV) which is a potent inhibitor of Hepatitis C Virus (HCV) NS5B polymerase. |
申请公布号 |
PT2084174(E) |
申请公布日期 |
2013.10.08 |
申请号 |
PT20070839369T |
申请日期 |
2007.10.05 |
申请人 |
F. HOFFMANN-LA ROCHE AG;GILEAD PHARMASSET LLC |
发明人 |
KESHAB SARMA;QINGWU JIN;BYOUNG-KWON CHUN;STEVEN D. AXT;JUSTIN VITALE;JIANG ZHU;BRUCE ROSS;SUGUNA RACHAKONDA |
分类号 |
C07H19/06;C07H5/02 |
主分类号 |
C07H19/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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