发明名称 Aminopyrimidines as SYK inhibitors
摘要 The present invention provides novel pyrimidine amines of formula (I) which are potent inhibitors of spleen tyrosine kinase, and are useful in the treatment and prevention of diseases mediated by said enzyme, such as asthma, COPD and rheumatoid arthritis.
申请公布号 US8551984(B2) 申请公布日期 2013.10.08
申请号 US20100968608 申请日期 2010.12.15
申请人 ALTMAN MICHAEL D.;ANDRESEN BRIAN M.;ARRINGTON KENNETH L.;BURCH JASON;CHILDERS KALEEN KONRAD;COTE BERNARD;DI FRANCESCO MARIA EMILIA;DONOFRIO ANTHONY;DUPONT-GAUDET KRISTINA;ELLIS JOHN MICHAEL;FISCHER CHRISTIAN;GUAY DANIEL;GUERIN DAVID JOSEPH;HAIDLE ANDREW M.;KATTAR SOLOMON;KNOWLES SANDRA LEE;LI CHAOMIN;LIM JONGWON;MACHACEK MICHELLE R.;NORTHRUP ALAN B.;O'BOYLE BRENDAN M.;OTTE RYAN D.;REUTERSHAN MICHAEL H.;ROMEO ERIC;SCHELL ADAM J.;SIU TONY;SPENCER KERRIE B.;TAOKA BRANDON M.;TROTTER B. WESLEY;ZHOU HUA;MERCK SHARP & DOHME CORP.;MERCK CANADA INC. 发明人 ALTMAN MICHAEL D.;ANDRESEN BRIAN M.;ARRINGTON KENNETH L.;BURCH JASON;CHILDERS KALEEN KONRAD;COTE BERNARD;DI FRANCESCO MARIA EMILIA;DONOFRIO ANTHONY;DUPONT-GAUDET KRISTINA;ELLIS JOHN MICHAEL;FISCHER CHRISTIAN;GUAY DANIEL;GUERIN DAVID JOSEPH;HAIDLE ANDREW M.;KATTAR SOLOMON;KNOWLES SANDRA LEE;LI CHAOMIN;LIM JONGWON;MACHACEK MICHELLE R.;NORTHRUP ALAN B.;O'BOYLE BRENDAN M.;OTTE RYAN D.;REUTERSHAN MICHAEL H.;ROMEO ERIC;SCHELL ADAM J.;SIU TONY;SPENCER KERRIE B.;TAOKA BRANDON M.;TROTTER B. WESLEY;ZHOU HUA
分类号 C07D417/12;A61K31/497 主分类号 C07D417/12
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