发明名称 DIPHENYL SULFIDE DERIVATIVE AND PHARMACEUTICAL PRODUCT WHICH CONTAINS SAME AS ACTIVE INGREDIENT
摘要 [Problem] To provide a diphenyl sulfide derivative which is useful as a pharmaceutical product that has excellent S1P3 antagonist activity. [Solution] The inventors have discovered that a diphenyl sulfide derivative represented by general formula (1) (wherein R1 represents an alkoxy group having 1-6 carbon atoms, R2 represents a propyl group or an allyl group, X represents methylene or an oxygen atom, and Z represents a halogen atom) has excellent S1P3 antagonist activity as a result of extensive researches for the production of a compound that has S1P3 antagonist activity.
申请公布号 US2013261089(A1) 申请公布日期 2013.10.03
申请号 US201113883847 申请日期 2011.12.20
申请人 ISHIKAWA KUMI;KOGA SHIGERU;KOHNO YASUSHI;FUJII KIYOSHI;YOSHIKAWA KEN 发明人 ISHIKAWA KUMI;KOGA SHIGERU;KOHNO YASUSHI;FUJII KIYOSHI;YOSHIKAWA KEN
分类号 C07F9/38 主分类号 C07F9/38
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